Aprocitentan (Standard) [1103522-45-7]

Aprocitentan (Standard) [1103522-45-7] : Size : 1L - Certification : Research Use Only - Aprocitentan (Standard) is the analytical standard of Aprocitentan. This product is intended for research and analytical applications. Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively[1]. -